...We Welcome You To The Resverlogix HUB withIn The AGORACOM COMMUNITY!

Free
Message: Bromodomain-2 Selective BET inhibitors

Imtesty,

Yes, I will post the links for the BD2-selective BET inhibitors and for Framework for Addressing Residual CVD risk to the link library. From what I understand, the BD2-selective compounds described in that paper, including apabetalone, are not selective for the BRD4 protein but also bind to others including BRD2 and BRD3 (possibly others, I don't know). Picaud et al documented this for apabetalone in this PNAS paper.

BearDownAZ

Share
New Message
Please login to post a reply